TRPV2 antagonist SET2 | TRPV2 antagonist | Probechem Biochemicals

Chemical Structure : TRPV2 antagonist SET2

CAS No.: 2313525-20-9

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TRPV2 antagonist SET2 (SET2)

货号: PC-22170Not For Human Use, Lab Use Only.

SET2 is a potent, subtype-selective inhibitor of transient receptor potential vanilloid type 2 (TRPV2) with IC50 of 0.46 uM.

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10 mg	￥1480	In stock
25 mg	￥2580	In stock
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生物&药学活性

SET2 is a potent, subtype-selective inhibitor of transient receptor potential vanilloid type 2 (TRPV2) with IC50 of 0.46 uM.
SET2 displays no activity against TRPV1, TRPV3, or TRPV4.
SET2 (0-20 uM) inhibits the migration of prostate cancer cell PC-3M expressing TRPV2.

物理化学性质&存储条件

分子量	402.44
分子式	C17H21F3N4O2S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(Furan-2-ylmethyl)-3-((4-(methyl(propyl)amino)-6-(trifluoromethyl)pyrimidin-2-yl)thio)propanamide

参考文献

1. Hao Chai, et al. J Med Chem. 2019 Feb 14;62(3):1373-1384.

TRPV2 antagonist SET2 (SET2)

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物理化学性质&存储条件

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TRPV2 antagonist SET2 (SET2)

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