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首页-小分子抑制剂&激动剂-Nuclear Receptor/Transcription Factor-RAR/RXR-LY-2955303
LY-2955303

Chemical Structure : LY-2955303

CAS No.: 1433497-19-8

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LY-2955303 (LY2955303)

货号: PC-62836Not For Human Use, Lab Use Only.

LY-2955303 is a potent and selective RARγ antagonist with binding Ki of 1.09 nM, displays >1000-fold selectivity against RARα and RARβ.

规格 价格 库存 数量
5 mg ￥980 In stock
10 mg ￥1480 In stock
25 mg ￥2580 In stock
50 mg ￥3980 In stock
100 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

LY-2955303 is a potent and selective RARγ antagonist with binding Ki of 1.09 nM, displays >1000-fold selectivity against RARα and RARβ.
LY-2955303 demonstrates good pharmacokinetic properties and efficacious in the MIA model of osteoarthritis-like joint pain.

物理化学性质&存储条件

分子量 578.76
分子式 C36H42N4O3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4-[5-[3,5-Bis(1,1-dimethylethyl)phenyl]-1-[4-[(4-methyl-1-piperazinyl)carbonyl]phenyl]-1H-pyrazol-3-yl]benzoic acid

参考文献

1. Hughes NE, et al. Bioorg Med Chem Lett. 2016 Jul 15;26(14):3274-7.

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