GSK-467 |CAS:1628332-52-4 Probechem Biochemicals

Chemical Structure : GSK-467

CAS No.: 1628332-52-4

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GSK-467 (GSK467, GSK 467)

货号: PC-62292Not For Human Use, Lab Use Only.

GSK-467 is a potent, selective KDM5 inhibitor with Ki of 10 nM, shows 180-fold selectivity for KDM4C and no measurable inhibitory effects toward KDM6 or other JmJ family members.

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5 mg	￥1580	In stock
10 mg	￥2480	In stock
25 mg	￥3980	In stock
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100 mg		Get quote

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生物&药学活性

GSK-467 (GSK467) is a potent, selective KDM5 inhibitor with Ki of 10 nM, shows 180-fold selectivity for KDM4C and no measurable inhibitory effects toward KDM6 or other JmJ family members.
GSK-467 (GSK467) increases the rate of apoptosis in myeloma cells.

物理化学性质&存储条件

分子量	319.32
分子式	C17H13N5O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-[(1-Benzyl-1H-pyrazol-4-yl)oxy]-pyrido-[3,4-d]pyrimidin-4(3H)-one

参考文献

1. Johansson C, et. Nat Chem Biol. 2016 Jul;12(7):539-45.

2. Westaway SM, et al. J Med Chem. 2016 Feb 25;59(4):1370-87.

GSK-467 (GSK467, GSK 467)

生物&药学活性

物理化学性质&存储条件

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GSK-467 (GSK467, GSK 467)

生物&药学活性

物理化学性质&存储条件

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