GSK-2879552 |CAS:1401966-69-5 Probechem Biochemicals

Chemical Structure : GSK-2879552

CAS No.: 1401966-69-5

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GSK-2879552 (GSK2879552)

货号: PC-45495Not For Human Use, Lab Use Only.

GSK-2879552 is a potent, selective irreversible inhibitor of LSD1 with Ki app of 1.7 uM.

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10 mg	￥1280	In stock
25 mg	￥1980	In stock
50 mg	￥2980	In stock
100 mg		Get quote

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生物&药学活性

GSK-2879552 is a potent, selective irreversible inhibitor of LSD1 with Ki app of 1.7 uM.
GSK-2879552 shows good selectivity against LSD2, MAO-A, MAO-B, D-amino acid oxidase and LoxL2.
GSK-2879552 exhibits growth inhibition (EC50=2-240 nM) in sensitive cell lines.
GSK-2879552 is orally bioavailable.

物理化学性质&存储条件

分子量	364.4806
分子式	C23H28N2O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Benzoic acid, 4-[[4-[[[(1R,2S)-2-phenylcyclopropyl]amino]methyl]-1-piperidinyl]methyl]-

参考文献

1. Mohammad HP, et al. Cancer Cell. 2015 Jul 13;28(1):57-69.

2. Huang M, et al. Cancer Lett. 2017 Jul 10;398:12-21.

3. Maes T, et al. Epigenomics. 2015;7(4):609-26.

GSK-2879552 (GSK2879552)

生物&药学活性

物理化学性质&存储条件

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GSK-2879552 (GSK2879552)

生物&药学活性

物理化学性质&存储条件

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