GSK-2140944 |CAS:1075236-89-3 Probechem Biochemicals

Chemical Structure : GSK-2140944

CAS No.: 1075236-89-3

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GSK-2140944 (Gepotidacin, GSK2140944)

货号: PC-61938Not For Human Use, Lab Use Only.

GSK-2140944 (Gepotidacin) is a novel potent, selective bacterial type II topoisomerase inhibitor in development for the treatment of conventional and biothreat pathogens, including Gram-positive pathogens and MRSA.

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5 mg	￥2980	In stock
10 mg	￥4780	In stock
25 mg	￥7280	In stock
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200 mg		Get quote
1 g		Get quote

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生物&药学活性

GSK-2140944 (Gepotidacin) is a novel potent, selective bacterial type II topoisomerase inhibitor in development for the treatment of conventional and biothreat pathogens, including Gram-positive pathogens and MRSA.
GSK-2140944 (Gepotidacin) shows antibacterial activity against MSSA and MRSA isolates (MIC90=0.5 ug/ml).

物理化学性质&存储条件

分子量	448.527
分子式	C24H28N6O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(2R)-2-[[4-[[(3,4-Dihydro-2H-pyrano[2,3-c]pyridin-6-yl)methyl]amino]-1-piperidinyl]methyl]-1,2-dihydro-3H,8H-2a,5,8a-triazaacenaphthylene-3,8-dione

参考文献

1. Bax BD, et al. Nature. 2010 Aug 19;466(7309):935-40.

2. Biedenbach DJ, et al. Antimicrob Agents Chemother. 2016 Jan 4;60(3):1918-23.

3. So W, et al. Antimicrob Agents Chemother. 2015 Aug;59(8):4956-61.

4. Farrell DJ, et al. Antimicrob Agents Chemother. 2017 Feb 23;61(3). pii: e02047-16.

GSK-2140944 (Gepotidacin, GSK2140944)

生物&药学活性

物理化学性质&存储条件

参考文献

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GSK-2140944 (Gepotidacin, GSK2140944)

生物&药学活性

物理化学性质&存储条件

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